BDBM265503 US9718808, 35

SMILES C[C@H]1C[C@]2(CC[C@@H](CC2)NCc2ccc(nn2)-n2cnnn2)C(=O)N1C1=CC(=O)OC1

InChI Key InChIKey=LJIZMRDHQSOIKQ-PJSUUKDQSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 265503   

TargetATP-sensitive inward rectifier potassium channel 1(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM265503(US9718808, 35)
Affinity DataIC50:  8.40nMAssay Description:A Thallium Flux Assay was performed on each of the final product compounds of the Examples. This assay has been described previously; see, e.g., PCT ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent